Page last updated: 2024-09-03

celastrol and 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione

celastrol has been researched along with 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione in 1 studies

Compound Research Comparison

Studies
(celastrol)
Trials
(celastrol)
Recent Studies (post-2010)
(celastrol)
Studies
(1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione)
Trials
(1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione)
Recent Studies (post-2010) (1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione)
88517411204

Protein Interaction Comparison

ProteinTaxonomycelastrol (IC50)1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione (IC50)
MPI proteinHomo sapiens (human)6.088
Apoptotic peptidase activating factor 1Homo sapiens (human)0.0375
caspase-9 isoform alpha precursorHomo sapiens (human)0.0256
sphingosine 1-phosphate receptor 2Homo sapiens (human)1.338
caspase-3 isoform a preproproteinHomo sapiens (human)0.0256
mothers against decapentaplegic homolog 3 isoform 1Homo sapiens (human)0.038
cysteine protease ATG4B isoform aHomo sapiens (human)3.73
tyrosine-protein phosphatase non-receptor type 22 isoform 1Homo sapiens (human)1.24
tyrosine-protein phosphatase non-receptor type 7 isoform 2Homo sapiens (human)1.24
RNA-editing ligase 1, mitochondrialTrypanosoma brucei brucei0.4108

Research

Studies (1)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's1 (100.00)2.80

Authors

AuthorsStudies
Li, L; Wang, L; Xu, XL; You, QD1

Reviews

1 review(s) available for celastrol and 1,3,6-trimethylpyrimido[5,4-e][1,2,4]triazine-5,7-dione

ArticleYear
Heat Shock Protein 90 Inhibitors: An Update on Achievements, Challenges, and Future Directions.
    Journal of medicinal chemistry, 2020, 03-12, Volume: 63, Issue:5

    Topics: Animals; Antineoplastic Agents; Autoimmune Diseases; Benzoquinones; Forecasting; HSP90 Heat-Shock Proteins; Humans; Immunosuppressive Agents; Lactams, Macrocyclic; Molecular Chaperones; Neoplasms; Protein Binding; Protein Structure, Secondary; Protein Structure, Tertiary

2020